No Cover Image

Journal article 986 views

Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation

Salvatore Ferla Orcid Logo, Mohamed S. Gomaa, Andrea Brancale, Jinge Zhu, Justin T. Ochalek, Hector F. DeLuca, Claire Simons

European Journal of Medicinal Chemistry, Volume: 87, Pages: 39 - 51

Swansea University Author: Salvatore Ferla Orcid Logo

Full text not available from this repository: check for access using links below.

Check full text

DOI (Published version): 10.1016/j.ejmech.2014.09.035

Published in: European Journal of Medicinal Chemistry
ISSN: 0223-5234
Published: Elsevier BV 2014
Online Access: Check full text

URI: https://cronfa.swan.ac.uk/Record/cronfa55495
first_indexed 2020-10-23T08:07:51Z
last_indexed 2020-12-11T04:19:47Z
id cronfa55495
recordtype SURis
fullrecord <?xml version="1.0"?><rfc1807><datestamp>2020-12-10T12:08:29.7750369</datestamp><bib-version>v2</bib-version><id>55495</id><entry>2020-10-22</entry><title>Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation</title><swanseaauthors><author><sid>d4c62248f510e3b221916989a7bbe6a6</sid><ORCID>0000-0002-5918-9237</ORCID><firstname>Salvatore</firstname><surname>Ferla</surname><name>Salvatore Ferla</name><active>true</active><ethesisStudent>false</ethesisStudent></author></swanseaauthors><date>2020-10-22</date><deptcode>MEDS</deptcode><abstract/><type>Journal Article</type><journal>European Journal of Medicinal Chemistry</journal><volume>87</volume><journalNumber/><paginationStart>39</paginationStart><paginationEnd>51</paginationEnd><publisher>Elsevier BV</publisher><placeOfPublication/><isbnPrint/><isbnElectronic/><issnPrint>0223-5234</issnPrint><issnElectronic/><keywords>Imidazole styrylindoles; Sulfonyl styrylindoles; CYP24A1; Vitamin D; Molecular modelling</keywords><publishedDay>24</publishedDay><publishedMonth>11</publishedMonth><publishedYear>2014</publishedYear><publishedDate>2014-11-24</publishedDate><doi>10.1016/j.ejmech.2014.09.035</doi><url/><notes/><college>COLLEGE NANME</college><department>Medical School</department><CollegeCode>COLLEGE CODE</CollegeCode><DepartmentCode>MEDS</DepartmentCode><institution>Swansea University</institution><apcterm/><lastEdited>2020-12-10T12:08:29.7750369</lastEdited><Created>2020-10-22T18:32:16.4268896</Created><path><level id="1">Faculty of Medicine, Health and Life Sciences</level><level id="2">Swansea University Medical School - Medicine</level></path><authors><author><firstname>Salvatore</firstname><surname>Ferla</surname><orcid>0000-0002-5918-9237</orcid><order>1</order></author><author><firstname>Mohamed S.</firstname><surname>Gomaa</surname><order>2</order></author><author><firstname>Andrea</firstname><surname>Brancale</surname><order>3</order></author><author><firstname>Jinge</firstname><surname>Zhu</surname><order>4</order></author><author><firstname>Justin T.</firstname><surname>Ochalek</surname><order>5</order></author><author><firstname>Hector F.</firstname><surname>DeLuca</surname><order>6</order></author><author><firstname>Claire</firstname><surname>Simons</surname><order>7</order></author></authors><documents/><OutputDurs/></rfc1807>
spelling 2020-12-10T12:08:29.7750369 v2 55495 2020-10-22 Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation d4c62248f510e3b221916989a7bbe6a6 0000-0002-5918-9237 Salvatore Ferla Salvatore Ferla true false 2020-10-22 MEDS Journal Article European Journal of Medicinal Chemistry 87 39 51 Elsevier BV 0223-5234 Imidazole styrylindoles; Sulfonyl styrylindoles; CYP24A1; Vitamin D; Molecular modelling 24 11 2014 2014-11-24 10.1016/j.ejmech.2014.09.035 COLLEGE NANME Medical School COLLEGE CODE MEDS Swansea University 2020-12-10T12:08:29.7750369 2020-10-22T18:32:16.4268896 Faculty of Medicine, Health and Life Sciences Swansea University Medical School - Medicine Salvatore Ferla 0000-0002-5918-9237 1 Mohamed S. Gomaa 2 Andrea Brancale 3 Jinge Zhu 4 Justin T. Ochalek 5 Hector F. DeLuca 6 Claire Simons 7
title Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
spellingShingle Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
Salvatore Ferla
title_short Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_full Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_fullStr Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_full_unstemmed Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
title_sort Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation
author_id_str_mv d4c62248f510e3b221916989a7bbe6a6
author_id_fullname_str_mv d4c62248f510e3b221916989a7bbe6a6_***_Salvatore Ferla
author Salvatore Ferla
author2 Salvatore Ferla
Mohamed S. Gomaa
Andrea Brancale
Jinge Zhu
Justin T. Ochalek
Hector F. DeLuca
Claire Simons
format Journal article
container_title European Journal of Medicinal Chemistry
container_volume 87
container_start_page 39
publishDate 2014
institution Swansea University
issn 0223-5234
doi_str_mv 10.1016/j.ejmech.2014.09.035
publisher Elsevier BV
college_str Faculty of Medicine, Health and Life Sciences
hierarchytype
hierarchy_top_id facultyofmedicinehealthandlifesciences
hierarchy_top_title Faculty of Medicine, Health and Life Sciences
hierarchy_parent_id facultyofmedicinehealthandlifesciences
hierarchy_parent_title Faculty of Medicine, Health and Life Sciences
department_str Swansea University Medical School - Medicine{{{_:::_}}}Faculty of Medicine, Health and Life Sciences{{{_:::_}}}Swansea University Medical School - Medicine
document_store_str 0
active_str 0
published_date 2014-11-24T04:51:19Z
_version_ 1851095546347913216
score 11.089407

Similar Items